Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
IC50: 100nMAssay Description:Inhibition of KDM5B in human ZR-75-1 cells assessed as reduction in H3K4me3 demethylation incubated for 72 hrs by fluorometric immunoassayMore data for this Ligand-Target Pair
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
IC50: 100nMAssay Description:Inhibition of KDM5A in human ZR-75-1 cells assessed as reduction in H3K4me3 demethylation incubated for 72 hrs by fluorometric immunoassayMore data for this Ligand-Target Pair
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
BDBM50158703(CHEMBL3785832 | US10173996, Example 53 | US9604961...)
EC50: 420nMAssay Description:Inhibition of KDM5A/KDM5B in human ZR-75-1 cells assessed as increase in H3K4me3 level after 72 hrs by fluorometric immunoassayMore data for this Ligand-Target Pair