Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetEgl nine homolog 1(Homo sapiens (Human))
TBA

Curated by ChEMBL

LigandBDBM50418048(CHEMBL1688408 | US10851083, Example 129 | US116187...)Copy SMILESCopy InChI

Affinity DataIC50:  100nMAssay Description:Inhibition of PHD2More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetEgl nine homolog 1 [181-417](Homo sapiens (Human))
Janssen Pharmaceutica

US Patent

LigandBDBM50418048(CHEMBL1688408 | US10851083, Example 129 | US116187...)Copy SMILESCopy InChI

Affinity DataIC50:  100nMAssay Description:The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetEgl nine homolog 1 [181-417](Homo sapiens (Human))
Janssen Pharmaceutica

US Patent

LigandBDBM50418048(CHEMBL1688408 | US10851083, Example 129 | US116187...)Copy SMILESCopy InChI

Affinity DataIC50:  100nMAssay Description:The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI