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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Tyrosine-protein kinase ZAP-70
(Homo sapiens (Human))
Ariad Pharmaceuticals
Ligand
BDBM5104
(1,2,4-Oxadiazole Analogue 15a | 4-[(2S)-2-{[(1S)-2...)
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Affinity Data
IC50: 3.00E+3nM
Assay Description:
Fluorescence polarization competitive binding assays were used to measure the IC50s of compounds binding to the different SH2 domains. The difference...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human))
Ariad Pharmaceuticals
Ligand
BDBM5104
(1,2,4-Oxadiazole Analogue 15a | 4-[(2S)-2-{[(1S)-2...)
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Affinity Data
IC50: 1.61E+5nM
Assay Description:
Fluorescence polarization competitive binding assays were used to measure the IC50s of compounds binding to the different SH2 domains. The difference...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase SYK
(Homo sapiens (Human))
Ariad Pharmaceuticals
Ligand
BDBM5104
(1,2,4-Oxadiazole Analogue 15a | 4-[(2S)-2-{[(1S)-2...)
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Copy InChI
Affinity Data
IC50: 3.18E+5nM
Assay Description:
Fluorescence polarization competitive binding assays were used to measure the IC50s of compounds binding to the different SH2 domains. The difference...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Growth factor receptor-bound protein 2
(Homo sapiens (Human))
Ariad Pharmaceuticals
Ligand
BDBM5104
(1,2,4-Oxadiazole Analogue 15a | 4-[(2S)-2-{[(1S)-2...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >5.00E+5nM
Assay Description:
Fluorescence polarization competitive binding assays were used to measure the IC50s of compounds binding to the different SH2 domains. The difference...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI