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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
Universite De Lyon
Ligand
BDBM34110
(glucopyranosylidene-spiro-isoxazoline, 4e)
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Affinity Data
Ki: 630nM ΔG°: -36.0kJ/mole
pH: 6.8 T: 2°C
Assay Description:
Phosphorylase activity was measured in the direction of glycogen synthesis by the release of orthophosphate from Glc-1-P. The enzyme was assayed in g...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
Universite De Lyon
Ligand
BDBM34110
(glucopyranosylidene-spiro-isoxazoline, 4e)
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Affinity Data
IC50: 630nM
Assay Description:
Binding affinity to rabbit muscular GPb by NMR binding assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glycogen phosphorylase, liver form
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM34110
(glucopyranosylidene-spiro-isoxazoline, 4e)
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Affinity Data
IC50: 1.42E+4nM
Assay Description:
Inhibition of glycogen phosphorylase in human hepatocytes assessed as glucagon stimulated glycogen content after 3 hrs by colorimetric GOD method
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, liver form
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM34110
(glucopyranosylidene-spiro-isoxazoline, 4e)
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Copy InChI
Affinity Data
IC50: 2.00E+4nM
Assay Description:
Inhibition of glycogen phosphorylase in human hepatocytes assessed as decrease in glucagon stimulated glucose release after 3 hrs by glucose oxidase ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, liver form
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM34110
(glucopyranosylidene-spiro-isoxazoline, 4e)
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Affinity Data
IC50: 3.60E+4nM
Assay Description:
Inhibition of glycogen phosphorylase in Wistar rat hepatocytes assessed as decrease in glucagon stimulated glucose release after 3 hrs by glucose oxi...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI