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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
18
hits in this display
Target
Lipopolysaccharide heptosyltransferase 1
(Escherichia coli (strain K12))
Wesleyan University
Curated by
ChEMBL
Ligand
BDBM34103
(D-glucose | dextrose | glucose)
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Affinity Data
Ki: 2.80E+5nM
Assay Description:
Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...
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Target
Glycogen phosphorylase, muscle form
(Homo sapiens (Human))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
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Affinity Data
Ki: 1.70E+6nM
Assay Description:
Inhibition of glycogen phosphorylase b (unknown origin)
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Target Info
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Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
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Affinity Data
Ki: 1.70E+6nM
Assay Description:
Competitive inhibition of rabbit skeletal muscle glycogen phosphorylase b using Glc-1-P as substrate
More data for this Ligand-Target Pair
Target Info
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PubMed
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Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.70E+6nM
Assay Description:
Inhibition of rabbit muscle glycogen phosphorylase inactive form b
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
KEGG
MMDB
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PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.70E+6nM
Assay Description:
Inhibition of rabbit muscle glycogen phosphorylase-b after 1 min in presence of varying levels of glucose-1-phosphate and constant concentration of g...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
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ChEBI
CHEMBL
KEGG
MMDB
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PC sid
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In Depth
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Article
PubMed
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Target
Glycogen phosphorylase, brain form
(Homo sapiens (Human))
University Of Perugia
Curated by
ChEMBL
Ligand
BDBM34103
(D-glucose | dextrose | glucose)
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Copy InChI
Affinity Data
Ki: 1.70E+6nM
Assay Description:
Inhibition of rabbit glycogen phosphorylase B enzyme
More data for this Ligand-Target Pair
Target Info
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Reactome pathway
KEGG
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antibodypedia
GoogleScholar
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ChEBI
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MMDB
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.70E+6nM
pH: 6.8
Assay Description:
Competitive inhibition of rabbit muscle glycogen phosphorylase b assessed as inorganic phosphate release using alphaD glucose-1-phosphate as substrat...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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ChEBI
CHEMBL
KEGG
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.00E+6nM
Assay Description:
Competitive inhibition of rabbit muscle glycogen phosphorylase-a in presence of varying levels of glucose-1-phosphate and constant concentration of g...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
KEGG
MMDB
PC cid
PC sid
Patents
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, muscle form
(Homo sapiens (Human))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM34103
(D-glucose | dextrose | glucose)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.77E+6nM
Assay Description:
Inhibitory activity against rabbit muscle glycogen phosphorylase
Checked by Author
More data for this Ligand-Target Pair
Target Info
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KEGG
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ChEBI
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Article
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PDB
3D Structure (crystal)
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Target
Glycogen phosphorylase, liver form
(Homo sapiens (Human))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
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Affinity Data
Ki: 4.28E+6nM
Assay Description:
Competitive inhibition of His6-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inorg...
More data for this Ligand-Target Pair
Target Info
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KEGG
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antibodypedia
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ChEBI
CHEMBL
KEGG
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PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, liver form
(Homo sapiens (Human))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50351158
(CHEMBL423707)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4.90E+6nM
Assay Description:
Inhibition of glycogen phosphorylase a (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
KEGG
MMDB
PC cid
PC sid
Patents
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, brain form
(Homo sapiens (Human))
University Of Perugia
Curated by
ChEMBL
Ligand
BDBM34103
(D-glucose | dextrose | glucose)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.40E+6nM
Assay Description:
Inhibitory binding constant against glycogen phosphorylase B
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
KEGG
MMDB
PC cid
PC sid
PDB
Patents
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, muscle form
(Oryctolagus cuniculus (rabbit))
University Of Thessaly
Curated by
ChEMBL
Ligand
BDBM50240803
(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.40E+6nM
Assay Description:
Inhibition of rabbit muscle glycogen phosphorylase inactive form b
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
KEGG
MMDB
PC cid
PC sid
PDB
Patents
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, brain form
(Homo sapiens (Human))
University Of Perugia
Curated by
ChEMBL
Ligand
BDBM34103
(D-glucose | dextrose | glucose)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.40E+6nM
Assay Description:
Inhibitory activity against muscle Glycogen Phosphorylase b
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
KEGG
MMDB
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, brain form
(Homo sapiens (Human))
University Of Perugia
Curated by
ChEMBL
Ligand
BDBM34103
(D-glucose | dextrose | glucose)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.94E+6nM
Assay Description:
Inhibitory activity against Pig Skeletal Glycogen Phosphorylase b
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
KEGG
MMDB
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycogen phosphorylase, brain form
(Homo sapiens (Human))
University Of Perugia
Curated by
ChEMBL
Ligand
BDBM34103
(D-glucose | dextrose | glucose)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.94E+6nM
Assay Description:
Inhibitory activity against Pig Skeletal Glycogen Phosphorylase b
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
KEGG
MMDB
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PC sid
PDB
Patents
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Asialoglycoprotein receptor 1
(Homo sapiens (Human))
University Of Basel
Curated by
ChEMBL
Ligand
BDBM50240803
(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
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Affinity Data
IC50: >3.00E+7nM
Assay Description:
Inhibition of D-GalNAc-PAA binding to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by competitive sol...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
KEGG
MMDB
PC cid
PC sid
PDB
Patents
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Asialoglycoprotein receptor 1
(Homo sapiens (Human))
University Of Basel
Curated by
ChEMBL
Ligand
BDBM50240803
(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Copy SMILES
Copy InChI
Affinity Data
Kd: >1.00E+7nM
Assay Description:
Binding affinity to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by surface plasmon resonance spectro...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
KEGG
MMDB
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI