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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 18 hits in this display   

TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  2.80E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition of glycogen phosphorylase b (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  1.70E+6nMAssay Description:Competitive inhibition of rabbit skeletal muscle glycogen phosphorylase b using Glc-1-P as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-b after 1 min in presence of varying levels of glucose-1-phosphate and constant concentration of g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition of rabbit glycogen phosphorylase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  1.70E+6nMpH: 6.8Assay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase b assessed as inorganic phosphate release using alphaD glucose-1-phosphate as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  2.00E+6nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-a in presence of varying levels of glucose-1-phosphate and constant concentration of g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  2.77E+6nMAssay Description:Inhibitory activity against rabbit muscle glycogen phosphorylaseChecked by AuthorMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  4.28E+6nMAssay Description:Competitive inhibition of His6-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inorg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50351158(CHEMBL423707)
Affinity DataKi:  4.90E+6nMAssay Description:Inhibition of glycogen phosphorylase a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  7.40E+6nMAssay Description:Inhibitory binding constant against glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University Of Thessaly

Curated by ChEMBL
LigandPNGBDBM50240803(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Affinity DataKi:  7.40E+6nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase inactive form bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  7.40E+6nMAssay Description:Inhibitory activity against muscle Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  7.94E+6nMAssay Description:Inhibitory activity against Pig Skeletal Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM34103(D-glucose | dextrose | glucose)
Affinity DataKi:  7.94E+6nMAssay Description:Inhibitory activity against Pig Skeletal Glycogen Phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50240803(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Affinity DataIC50: >3.00E+7nMAssay Description:Inhibition of D-GalNAc-PAA binding to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by competitive sol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsialoglycoprotein receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50240803(CHEMBL1614854 | Glucoside | beta-D-glucopyranose |...)
Affinity DataKd: >1.00E+7nMAssay Description:Binding affinity to human recombinant ASGPR1 carbohydrate recognition domain expressed in Escherichia coli AD494 by surface plasmon resonance spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed