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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Fatty acid synthase
(Homo sapiens (Human))
Forma Therapeutics
Curated by
ChEMBL
Ligand
BDBM50526401
(CHEMBL4445590)
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Affinity Data
IC50: 61nM
Assay Description:
Inhibition of FASN in human BT474 cells preincubated for 1 hr followed by [14C]-acetate addition and measured after 4 hrs by scintillation counting a...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Fatty acid synthase
(Homo sapiens (Human))
Forma Therapeutics
Curated by
ChEMBL
Ligand
BDBM50526401
(CHEMBL4445590)
Copy SMILES
Copy InChI
Affinity Data
IC50: 192nM
Assay Description:
Inhibition of full length recombinant human FASN using acetyl-CoA/malonyl-CoA as substrate preincubated for 60 mins followed by substrate addition an...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI