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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Section De Chimie De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50104305(2-{[(Imidazol-1-ylmethyl)-amino]-methyl}-pyrrolidi...)
Affinity DataKi:  1.20E+5nMAssay Description:Inhibitory activity towards Beta-Glucosidase from Caldocellum saccharolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidase(Homo sapiens (Human))
Universidade Do Porto 687

Curated by ChEMBL
LigandPNGBDBM50402982(CHEMBL2207392)
Affinity DataKi:  3.26E+5nMAssay Description:Inhibition of human ER alpha mannosidase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-mannosidase 2(Homo sapiens (Human))
Universidade Do Porto 687

Curated by ChEMBL
LigandPNGBDBM50402982(CHEMBL2207392)
Affinity DataKi:  5.68E+5nMAssay Description:Inhibition of human golgi alpha mannosidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Section De Chimie De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50104305(2-{[(Imidazol-1-ylmethyl)-amino]-methyl}-pyrrolidi...)
Affinity DataIC50:  2.90E+5nMAssay Description:Inhibitory activity towards Alpha-glucosidase from Aspergillus niger (amyloglucosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucosidase(Prunus avium)
Section De Chimie De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50104305(2-{[(Imidazol-1-ylmethyl)-amino]-methyl}-pyrrolidi...)
Affinity DataIC50:  4.20E+5nMAssay Description:Inhibitory activity towards Beta-Glucosidase from AlmondMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetalpha-1,2-Mannosidase(Glycine max)
Section De Chimie De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50104305(2-{[(Imidazol-1-ylmethyl)-amino]-methyl}-pyrrolidi...)
Affinity DataIC50:  5.70E+5nMAssay Description:Inhibitory activity towards Alpha-mannosidase from AlmondMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetalpha-1,2-Mannosidase(Glycine max)
Section De Chimie De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50104305(2-{[(Imidazol-1-ylmethyl)-amino]-methyl}-pyrrolidi...)
Affinity DataIC50:  7.00E+5nMAssay Description:Inhibitory activity towards Beta-galactosidase from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed