Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMacrophage metalloelastase(Homo sapiens (Human))
Protera

Curated by ChEMBL
LigandPNGBDBM50332951(2-(4-fluoro-N-(2-hydroxyethyl)phenylsulfonamido)-N...)
Affinity DataKi:  40nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCollagenase 3(Homo sapiens (Human))
Protera

Curated by ChEMBL
LigandPNGBDBM50332951(2-(4-fluoro-N-(2-hydroxyethyl)phenylsulfonamido)-N...)
Affinity DataKi:  46nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Protera

Curated by ChEMBL
LigandPNGBDBM50332951(2-(4-fluoro-N-(2-hydroxyethyl)phenylsulfonamido)-N...)
Affinity DataKi:  151nMAssay Description:Inhibition of MMP1 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Protera

Curated by ChEMBL
LigandPNGBDBM50332951(2-(4-fluoro-N-(2-hydroxyethyl)phenylsulfonamido)-N...)
Affinity DataKi:  173nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Protera

Curated by ChEMBL
LigandPNGBDBM50332951(2-(4-fluoro-N-(2-hydroxyethyl)phenylsulfonamido)-N...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of MMP7 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed