Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant full-length human PKCtheta using STK1-biotin as substrate preincubated for 60 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50517664(CHEMBL4526554)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human full length PKCtheta using biotin-labelled STK substrate-1 as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of PKCtheta in human Jurkat cells transfected with pGL3-IL2 pro 43 plasmid assessed as suppression of IL-2 production after 14 hrs by fire...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCepsilon expressed in Baculovirus expression system using STK1-biotin as substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCdelta expressed in Baculovirus expression system using STK1-biotin as substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  84nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCalpha expressed in Baculovirus expression system using STK1-biotin as substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50: >300nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCeta expressed in Baculovirus expression system using STK1-biotin as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50:  410nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCbeta1 expressed in Baculovirus expression system using STK1-biotin as substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCzeta expressed in Baculovirus expression system using STK1-biotin as substrate af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50469246(CHEMBL4289707)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant N-terminal GST-fused full-length human PKCgamma expressed in Baculovirus expression system using STK1-biotin as substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed