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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099465((R)-1-[4-(4-Fluoro-phenoxy)-benzyl]-2-oxo-imidazol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Matrix metalloproteinase-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099465((R)-1-[4-(4-Fluoro-phenoxy)-benzyl]-2-oxo-imidazol...)
Affinity DataIC50:  28nMAssay Description:Inhibition of Matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099465((R)-1-[4-(4-Fluoro-phenoxy)-benzyl]-2-oxo-imidazol...)
Affinity DataIC50:  62nMAssay Description:Inhibition of Matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099465((R)-1-[4-(4-Fluoro-phenoxy)-benzyl]-2-oxo-imidazol...)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099465((R)-1-[4-(4-Fluoro-phenoxy)-benzyl]-2-oxo-imidazol...)
Affinity DataIC50:  5.45E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed