Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099466((R)-1-[4-(Naphthalen-2-yloxy)-benzyl]-2-oxo-imidaz...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Matrix metalloproteinase-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099466((R)-1-[4-(Naphthalen-2-yloxy)-benzyl]-2-oxo-imidaz...)
Affinity DataIC50:  56nMAssay Description:Inhibition of Matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099466((R)-1-[4-(Naphthalen-2-yloxy)-benzyl]-2-oxo-imidaz...)
Affinity DataIC50:  59nMAssay Description:Inhibition of Matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099466((R)-1-[4-(Naphthalen-2-yloxy)-benzyl]-2-oxo-imidaz...)
Affinity DataIC50:  940nMAssay Description:Inhibition of Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50099466((R)-1-[4-(Naphthalen-2-yloxy)-benzyl]-2-oxo-imidaz...)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed