Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 17 hits in this display
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
Ki: >4.50E+3nMAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
Matrilysin(Homo sapiens (Human))Bristol-Myers Squibb
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
Ki: >6.37E+3nMAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
Matrilysin(Homo sapiens (Human))Bristol-Myers Squibb
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)
BDBM26575((3R,4R)-3-N-hydroxy-4-N-(4-{[2-(trifluoromethyl)py...)