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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetPyruvate kinase PKLR(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50143419(CHEMBL175336 | Sodium; 3,4-dihydroxy-9,10-dioxo-9,...)
Affinity DataIC50:  200nMAssay Description:Inhibition of PKL (unknown origin) for 30 mins by Kinase-Glo Max reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhosphoglycerate mutase 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50143419(CHEMBL175336 | Sodium; 3,4-dihydroxy-9,10-dioxo-9,...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of PGAM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Inha University

Curated by ChEMBL
LigandPNGBDBM50143419(CHEMBL175336 | Sodium; 3,4-dihydroxy-9,10-dioxo-9,...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of human PTPase 1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase 1(Saccharomyces cerevisiae)
Inha University

Curated by ChEMBL
LigandPNGBDBM50143419(CHEMBL175336 | Sodium; 3,4-dihydroxy-9,10-dioxo-9,...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibitory activity against Saccharomyces cerevisiae Tyrosine phosphatase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed