Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50236545(CHEMBL4087125)
Affinity DataIC50:  42nMAssay Description:Antagonistic activity against human androgen receptor (hAR) in CV-1 cells using cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50236545(CHEMBL4087125)
Affinity DataIC50:  86nMAssay Description:Inhibition of DYRK1A (unknown origin) using woodtide as substrate after 10 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50236545(CHEMBL4087125)
Affinity DataIC50:  408nMAssay Description:Inhibition of DYRK2 (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50236545(CHEMBL4087125)
Affinity DataEC50:  7.00E+4nMAssay Description:Antagonistic activity against human androgen receptor (hAR) in CV-1 cells using cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed