Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 19 hits in this display
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 2.10nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 2.30nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 3.70nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 4.30nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 4.40nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 4.60nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 5.10nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 17.7nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 21.6nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 25.2nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 26.1nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 50.7nMpH: 8.0Assay Description:The inhibitory activity measurement against the kinases mentioned above was measured in the kinase inhibition reaction mixture containing 2 ul purifi...More data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 164nMAssay Description:Inhibition of human DDR1b expressed in HEK293 cells assessed as reduction in collagen-1-induced receptor auto-phosphorylation by Western blot methodMore data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 164nMAssay Description:Inhibition of type 1 collagen-induced autophosphorylation of human recombinant DDR1 expressed in HEK293 cells by Western blotting analysisMore data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 171nMAssay Description:Inhibition of human DDR2 expressed in HEK293 cells assessed as reduction in collagen-1-induced receptor auto-phosphorylation by Western blot methodMore data for this Ligand-Target Pair
BDBM50430875(CHEMBL2336005 | US9062066, LCB 03-0110)
IC50: 171nMAssay Description:Inhibition of type 1 collagen-induced autophosphorylation of human recombinant DDR2 expressed in HEK293 cells by Western blotting analysisMore data for this Ligand-Target Pair