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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Curtin University

Curated by ChEMBL
LigandPNGBDBM50197065(CHEMBL3913354)
Affinity DataIC50:  2nMAssay Description:Inhibition of DNA-PK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50197065(CHEMBL3913354)
Affinity DataIC50:  8nMAssay Description:Inhibition of PI3Kalpha/p85alpha (unknown origin) using phosphatidylinositol and gamma-32P-ATP incubated for 20 mins by TLC assay or high-throughput ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Homo sapiens (Human))
Curtin University

Curated by ChEMBL
LigandPNGBDBM50197065(CHEMBL3913354)
Affinity DataIC50:  26nMAssay Description:Inhibition of PI3KC2beta (unknown origin) expressed in HEK293 cells using phosphatidylinositol and gamma-32P-ATP incubated for 20 mins by TLC assay o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha(Homo sapiens (Human))
Curtin University

Curated by ChEMBL
LigandPNGBDBM50197065(CHEMBL3913354)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of PI3KC2alpha (unknown origin) expressed in HEK293 cells using phosphatidylinositol and gamma-32P-ATP incubated for 20 mins by TLC assay ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Curtin University

Curated by ChEMBL
LigandPNGBDBM50197065(CHEMBL3913354)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human Vps34 assessed as reduction in lipid kinase activity using PV5122 substrate incubated for 1 hr by Adapta kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Curtin University

Curated by ChEMBL
LigandPNGBDBM50197065(CHEMBL3913354)
Affinity DataIC50:  2.30E+6nMAssay Description:Inhibition of full length human recombinant VPS34 (unknown origin) using phosphatidylinositol and gamma-32P-ATP incubated for 20 mins by TLC assay or...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed