Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 19 hits in this display
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
IC50: 4.36E+3nMAssay Description:The protocol for measuring IC50 values for the inhibition of MAO-A and MAO-B has been reported in detail in a recent publication (26). The recombinan...More data for this Ligand-Target Pair
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
IC50: 5.40E+3nMpH: 7.0 T: 2°CAssay Description:The enzymatic activities of FtFabZ and YpFabZ were determined via the reportedspectrophotometric method using the substrate analogue crotonoyl-CoA.7 ...More data for this Ligand-Target Pair
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
IC50: 1.01E+4nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-Pro-Phe-4-nitroanilide as substrate after 30 mins by protease-coupled assayMore data for this Ligand-Target Pair
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
IC50: 1.70E+4nMAssay Description:5-LO inhibitory activity was determined by inhibition of LTB4 biosynthesis in bovine polymorphonuclear leukocytes (PMNL)More data for this Ligand-Target Pair
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
EC50: 1.70E+3nMAssay Description:Activation of human TRPA1 expressed in HEK293 cells assessed as increase in calcium level by fluo-4 dye based plate reader analysisMore data for this Ligand-Target Pair
BDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | 5-hyd...)
EC50: 1.70E+3nMAssay Description:Activation of human TRPA1 expressed in HEK293 cells assessed as increase in calcium level by fluo-4 dye based plate reader analysisMore data for this Ligand-Target Pair