Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105913(CHEMBL3597991)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant GST-fused Dyrk2 expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105913(CHEMBL3597991)
Affinity DataIC50:  70nMAssay Description:Inhibition of human recombinant Dyrk1B using Woodtide as substrate after 15 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50105913(CHEMBL3597991)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant His6-tagged Dyrk1A expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed