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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kJ/mol
)
Found
13
hits in this display
Target
Norepinephrine transporter
(RAT)
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
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Affinity Data
Ki: 18nM
More data for this Ligand-Target Pair
Target Info
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 150nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 840nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M2
(RAT)
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4.70E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Transporter
(Rattus norvegicus)
TBA
Curated by
ChEMBL
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 18nM
Assay Description:
Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Transporter
(Rattus norvegicus)
TBA
Curated by
ChEMBL
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 40nM
Assay Description:
Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 150nM
Assay Description:
Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 210nM
Assay Description:
Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Transporter
(Rattus norvegicus)
TBA
Curated by
ChEMBL
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 370nM
Assay Description:
Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 840nM
Assay Description:
Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.40E+3nM
Assay Description:
Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.48E+3nM
Assay Description:
Inhibition of 5-HT uptake in synaptosomal preparation from rat corpus striatum, using [3H]5-HT
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
Pfizer
Curated by
PDSP K
i
Database
Ligand
BDBM82219
(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.40E+4nM
Assay Description:
Inhibition of 5-HT uptake in synaptosomal preparation from rat corpus striatum, using [3H]5-HT
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI