Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 140 hits in this display   

TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  2nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  2nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  3nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  3nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  4nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  6nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313797(US10167292, Example 41)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313807(US10167292, Example 51B)
Affinity DataIC50:  7nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  9nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313796(US10167292, Example 40)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  10nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313803(US10167292, Example 47)
Affinity DataIC50:  11nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  11nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313777(US10167292, Example 12)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313771(US10167292, Example 5)
Affinity DataIC50:  12nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313803(US10167292, Example 47)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313797(US10167292, Example 41)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  13nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313777(US10167292, Example 12)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313794(US10167292, Example 38)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  14nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  15nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313793(US10167292, Example 37)
Affinity DataIC50:  15nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313788(US10167292, Example 32)
Affinity DataIC50:  16nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  16nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  16nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313788(US10167292, Example 32)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285938(CHEMBL4174918)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  17nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313787(US10167292, Example 31)
Affinity DataIC50:  18nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  18nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313787(US10167292, Example 31)
Affinity DataIC50:  18nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313771(US10167292, Example 5)
Affinity DataIC50:  19nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  19nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  20nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285938(CHEMBL4174918)
Affinity DataIC50:  21nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  21nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  21nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313793(US10167292, Example 37)
Affinity DataIC50:  21nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313796(US10167292, Example 40)
Affinity DataIC50:  21nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313796(US10167292, Example 40)
Affinity DataIC50:  21nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313777(US10167292, Example 12)
Affinity DataIC50:  23nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313806(US10167292, Example 50)
Affinity DataIC50:  23nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  23nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313803(US10167292, Example 47)
Affinity DataIC50:  24nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313776(US10167292, Example 11)
Affinity DataIC50:  25nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  25nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  25nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313797(US10167292, Example 41)
Affinity DataIC50:  25nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313796(US10167292, Example 40)
Affinity DataIC50:  25nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  26nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  28nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313788(US10167292, Example 32)
Affinity DataIC50:  28nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313771(US10167292, Example 5)
Affinity DataIC50:  28nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  28nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285938(CHEMBL4174918)
Affinity DataIC50:  29nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313787(US10167292, Example 31)
Affinity DataIC50:  29nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313790(US10167292, Example 34)
Affinity DataIC50:  30nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313776(US10167292, Example 11)
Affinity DataIC50:  32nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313774(US10167292, Example 8)
Affinity DataIC50:  33nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313798(US10167292, Example 42)
Affinity DataIC50:  34nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  34nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  34nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313776(US10167292, Example 11)
Affinity DataIC50:  35nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313775(US10167292, Example 10)
Affinity DataIC50:  35nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313793(US10167292, Example 37)
Affinity DataIC50:  35nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313781(US10167292, Example 21)
Affinity DataIC50:  36nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313790(US10167292, Example 34)
Affinity DataIC50:  36nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313793(US10167292, Example 37)
Affinity DataIC50:  37nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313780(US10167292, Example 20)
Affinity DataIC50:  38nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313779(US10167292, Example 16)
Affinity DataIC50:  38nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313777(US10167292, Example 12)
Affinity DataIC50:  38nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313771(US10167292, Example 5)
Affinity DataIC50:  39nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313794(US10167292, Example 38)
Affinity DataIC50:  39nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313790(US10167292, Example 34)
Affinity DataIC50:  40nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313776(US10167292, Example 11)
Affinity DataIC50:  43nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313806(US10167292, Example 50)
Affinity DataIC50:  43nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313781(US10167292, Example 21)
Affinity DataIC50:  44nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285938(CHEMBL4174918)
Affinity DataIC50:  44nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313797(US10167292, Example 41)
Affinity DataIC50:  44nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313794(US10167292, Example 38)
Affinity DataIC50:  44nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313794(US10167292, Example 38)
Affinity DataIC50:  44nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313781(US10167292, Example 21)
Affinity DataIC50:  45nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313780(US10167292, Example 20)
Affinity DataIC50:  45nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313788(US10167292, Example 32)
Affinity DataIC50:  50nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313791(US10167292, Example 35)
Affinity DataIC50:  51nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313787(US10167292, Example 31)
Affinity DataIC50:  52nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313781(US10167292, Example 21)
Affinity DataIC50:  52nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313780(US10167292, Example 20)
Affinity DataIC50:  52nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313778(US10167292, Example 13)
Affinity DataIC50:  53nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313773(US10167292, Example 7)
Affinity DataIC50:  53nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313796(US10167292, Example 40)
Affinity DataIC50:  54nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313803(US10167292, Example 47)
Affinity DataIC50:  56nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313777(US10167292, Example 12)
Affinity DataIC50:  64nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313795(US10167292, Example 39)
Affinity DataIC50:  68nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  77nMAssay Description:Inhibition of binding of a tetra-acetylated histone H4 peptide to His-tagged human BRD4(D1) expressed in bacteriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313790(US10167292, Example 34)
Affinity DataIC50:  79nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313792(US10167292, Example 36)
Affinity DataIC50:  79nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313789(US10167292, Example 33)
Affinity DataIC50:  95nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313787(US10167292, Example 31)
Affinity DataIC50:  116nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313776(US10167292, Example 11)
Affinity DataIC50:  129nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285938(CHEMBL4174918)
Affinity DataIC50:  129nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313793(US10167292, Example 37)
Affinity DataIC50:  136nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313780(US10167292, Example 20)
Affinity DataIC50:  147nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313794(US10167292, Example 38)
Affinity DataIC50:  151nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313788(US10167292, Example 32)
Affinity DataIC50:  185nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313806(US10167292, Example 50)
Affinity DataIC50:  204nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313771(US10167292, Example 5)
Affinity DataIC50:  264nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313780(US10167292, Example 20)
Affinity DataIC50:  273nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313781(US10167292, Example 21)
Affinity DataIC50:  340nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313806(US10167292, Example 50)
Affinity DataIC50:  370nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313790(US10167292, Example 34)
Affinity DataIC50:  388nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313772(US10167292, Example 6)
Affinity DataIC50: >999nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313772(US10167292, Example 6)
Affinity DataIC50: >999nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313772(US10167292, Example 6)
Affinity DataIC50: >999nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM313772(US10167292, Example 6)
Affinity DataIC50: >999nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285939(CHEMBL4160537)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285939(CHEMBL4160537)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285939(CHEMBL4160537)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285939(CHEMBL4160537)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter And Eliza Hall Institute Of Medical Research

Curated by ChEMBL
LigandPNGBDBM50285939(CHEMBL4160537)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed