Report error Found 3 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467]'
TargetGamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467](Human)
University of Wisconsin At Madison
University of Wisconsin At Madison
Affinity DataKi: 1.5nM ΔG°: -50.4kJ/moleT: 25°CAssay Description:Membrane homogenates were incubated at room temperature with a sub-Kd concentration of radioligand in the absence or presence of seven different conc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467](Human)
University of Wisconsin At Madison
University of Wisconsin At Madison
Affinity DataKi: 249nM ΔG°: -37.7kJ/moleT: 25°CAssay Description:Membrane homogenates were incubated at room temperature with a sub-Kd concentration of radioligand in the absence or presence of seven different conc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467](Human)
University of Wisconsin At Madison
University of Wisconsin At Madison
Affinity DataKi: 556nM ΔG°: -35.7kJ/moleT: 25°CAssay Description:Membrane homogenates were incubated at room temperature with a sub-Kd concentration of radioligand in the absence or presence of seven different conc...More data for this Ligand-Target Pair