Report error Found 135 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group D member 1'
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Agonist activity at Rev-Erbalpha expressed in HEK293 cells coexpressing Gal4 ligand binding domain assessed as inhibition of transcription after 24 h...More data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 710nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
Affinity DataKd: 800nMAssay Description:Dissociation constant for binding to REV-ERB-alpha by circular dichroismMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair