Report error Found 332 Enz. Inhib. hit(s) with Target = 'Endoplasmic reticulum aminopeptidase 1'
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 991nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.52E+3nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 2.54E+3nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of binding of [3H]citalopram to (SERT) serotonin transporter in rat striatumMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 3.73E+3nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Competitive inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using varying le...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 4.94E+3nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 5.08E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 5.55E+3nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 6.27E+3nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 6.47E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.09E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.13E+4nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.23E+4nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.28E+4nMAssay Description:Competitive inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using varying le...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.75E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.85E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.86E+4nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.91E+4nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 2.34E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 2.69E+4nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 3.16E+4nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 4.40E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 5.17E+4nMAssay Description:Competitive inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using varying le...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 8.71E+4nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 1.51E+5nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrateMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: 2.49E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric met...More data for this Ligand-Target Pair
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