Report error Found 654 Enz. Inhib. hit(s) with Target = 'Microtubule-associated protein tau'
Affinity DataKi: 0.180nM ΔG°: -55.6kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.220nM ΔG°: -55.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.224nM ΔG°: -55.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.290nM ΔG°: -54.4kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.290nM ΔG°: -54.4kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.320nM ΔG°: -54.2kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nM ΔG°: -54.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nM ΔG°: -54.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.383nM ΔG°: -53.7kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nM ΔG°: -53.6kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.410nM ΔG°: -53.6kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.423nM ΔG°: -53.5kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.430nM ΔG°: -53.5kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.430nM ΔG°: -53.5kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.438nM ΔG°: -53.4kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Displacement of [11C]PBB3 in human brain tau incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Displacement of Thioflavin S from recombinant human tau expressed in Escherichia coli after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nM ΔG°: -53.2kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.480nM ΔG°: -53.2kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.494nM ΔG°: -53.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.512nM ΔG°: -53.0kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.530nM ΔG°: -52.9kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.530nM ΔG°: -52.9kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.540nM ΔG°: -52.9kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.550nM ΔG°: -52.9kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.620nM ΔG°: -52.6kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.670nM ΔG°: -52.4kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.672nM ΔG°: -52.4kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.677nM ΔG°: -52.3kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.690nM ΔG°: -52.3kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.75nM ΔG°: -52.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.75nM ΔG°: -52.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.760nM ΔG°: -52.0kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.784nM ΔG°: -52.0kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.870nM ΔG°: -51.7kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.960nM ΔG°: -51.5kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 0.980nM ΔG°: -51.4kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.02nM ΔG°: -51.3kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.05nM ΔG°: -51.2kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.06nM ΔG°: -51.2kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.07nM ΔG°: -51.2kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.09nM ΔG°: -51.2kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.13nM ΔG°: -51.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.13nM ΔG°: -51.1kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.14nM ΔG°: -51.0kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.14nM ΔG°: -51.0kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.16nM ΔG°: -51.0kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.17nM ΔG°: -51.0kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.23nM ΔG°: -50.9kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
Affinity DataKi: 1.28nM ΔG°: -50.8kJ/molepH: 7.4 T: 25°CAssay Description:For displacement tau binding assay, unlabeled test compounds were dissolved in DMSO at 1 mM. Dilutions of tests compounds to various concentrations w...More data for this Ligand-Target Pair
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