Report error Found 116 Enz. Inhib. hit(s) with Target = 'Telomeric repeat-binding factor 2'
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.89E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 5.80E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 6.20E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 8.80E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 1.13E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 1.32E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 1.37E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataKi: 1.39E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
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