TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKi: 1.25E+4nMAssay Description:Competitive inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrateMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKi: 1.00E+5nMAssay Description:Inhibition of isopeptidase TMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of AChE in organophosphate-susceptible clone of Schizaphis graminum OSS adult or last-instar nymphs homogenates assessed as bimolecular ra...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of USP5 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of AChE in organophosphate-resistant clone of Schizaphis graminum OR1 adult or last-instar nymphs homogenates assessed as bimolecular rate...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human 6His-tagged USP5 expressed in Escherichia coli assessed as cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine1...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Ligand InfoPDB
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of AChE in organophosphate-susceptible clone of Schizaphis graminum OSS adult or last-instar nymphs homogenates assessed as bimolecular ra...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Ligand Info
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of AChE in organophosphate-resistant clone of Schizaphis graminum OR1 adult or last-instar nymphs homogenates assessed as bimolecular rate...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of USP5 (unknown origin) using Ub-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by fluor...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Ligand Info
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 9.40E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 1.50E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 5.40E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 9.00E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 9.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 8.70E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 6.10E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 1.30E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.20E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 8.00E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 3.80E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 4.50E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 3.40E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 1.50E+5nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.50E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 1.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 4.00E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.30E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.10E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 7.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 1.80E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 3.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 3.10E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 8.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 4.20E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 4.70E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 5.90E+4nMAssay Description:Inhibition of carbonic anhydrase 2 assessed as inhibition of carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 9.00E+3nMAssay Description:Binding affinity to human CD69 receptor expressed in Escherichia coli by equilibrium dialysisMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.10E+5nMAssay Description:Binding affinity to human monomeric CD69 receptor expressed in Escherichia coli by equilibrium dialysisMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to human dimeric CD69 receptor expressed in Escherichia coli by equilibrium dialysisMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 7.00E+3nMAssay Description:Inhibition of Manduca sexta V-ATPase V1/Vo holoenzyme activity assessed as inorganic phosphate production pretreated for 5 minsMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.20E+4nMAssay Description:Inhibition of Manduca sexta V-ATPase V1/Vo holoenzyme activity assessed as inorganic phosphate production pretreated for 5 minsMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 2.10E+4nMAssay Description:Inhibition of Manduca sexta V-ATPase V1/Vo holoenzyme activity assessed as inorganic phosphate production pretreated for 5 minsMore data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture
Curated by ChEMBL
Tokyo University Of Agriculture
Curated by ChEMBL
Affinity DataKd: 6.10E+4nMAssay Description:Inhibition of Manduca sexta V-ATPase V1/Vo holoenzyme activity assessed as inorganic phosphate production pretreated for 5 minsMore data for this Ligand-Target Pair