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Found 14 Enz. Inhib. hit(s) with Target = 'C-type lectin domain family 4 member K'
TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50608273(CHEMBL5271773)
Affinity DataKi:  3.20E+5nMAssay Description:Binding affinity to Langerin (unknown origin) by [19F] R2-filtered NMR assayMore data for this Ligand-Target Pair
Ligand Info
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50608271(CHEMBL5272018)
Affinity DataKi:  1.30E+6nMAssay Description:Binding affinity to Langerin (unknown origin) by [19F] R2-filtered NMR assayMore data for this Ligand-Target Pair
Ligand Info
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50608272(CHEBI:16702 | GLUCOSAMINE SULFATE)
Affinity DataKi:  1.40E+6nMAssay Description:Binding affinity to Langerin (unknown origin) by [19F] R2-filtered NMR assayMore data for this Ligand-Target Pair
Ligand Info
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50608270(CHEMBL5283516)
Affinity DataKi:  7.60E+6nMAssay Description:Binding affinity to Langerin (unknown origin) by [19F] R2-filtered NMR assayMore data for this Ligand-Target Pair
Ligand Info
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50608269(CHEMBL5286552)
Affinity DataKi:  4.80E+7nMAssay Description:Binding affinity to Langerin (unknown origin) by [19F] R2-filtered NMR assayMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50608274(CHEMBL5275954)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of mannan binding to mouse Langerin extracellular domain by ELLA assayMore data for this Ligand-Target Pair
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50610694(CHEMBL5289548)
Affinity DataIC50:  5.80E+5nMAssay Description:Inhibition of human Langerin overexpressed in human Raji cells incubated for 30 mins by flow cytometryMore data for this Ligand-Target Pair
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM85507(CAS_4394-00-7 | NSC_4488 | Niflumic acid | Niflumi...)
Affinity DataIC50:  5.90E+5nMAssay Description:Inhibition of human Langerin overexpressed in human Raji cells incubated for 30 mins by flow cytometryMore data for this Ligand-Target Pair
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50399360(CHEMBL1852052)
Affinity DataIC50:  1.00E+6nMAssay Description:Displacement of biotinylated-TM PAA from human langerin after 3 hrs by colorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50610690(CHEMBL5290361)
Affinity DataIC50:  1.03E+6nMAssay Description:Inhibition of human Langerin overexpressed in human Raji cells incubated for 30 mins by flow cytometryMore data for this Ligand-Target Pair
Ligand Info
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50610691(CHEMBL5269455)
Affinity DataIC50:  1.06E+6nMAssay Description:Inhibition of human Langerin overexpressed in human Raji cells incubated for 30 mins by flow cytometryMore data for this Ligand-Target Pair
Ligand Info
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50610692(CHEMBL5266266)
Affinity DataIC50:  1.15E+6nMAssay Description:Inhibition of human Langerin overexpressed in human Raji cells incubated for 30 mins by flow cytometryMore data for this Ligand-Target Pair
Ligand Info
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TargetC-type lectin domain family 4 member K(Homo sapiens (Human))TBA
LigandPNGBDBM50610693(CHEMBL5272727)
Affinity DataIC50:  1.19E+6nMAssay Description:Inhibition of human Langerin overexpressed in human Raji cells incubated for 30 mins by flow cytometryMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50608274(CHEMBL5275954)
Affinity DataKd:  4.50E+5nMAssay Description:Inhibition of mannan binding to mouse Langerin extracellular domain assessed as apparent dissociation constant by ELLA assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed