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Found 884 Enz. Inhib. hit(s) with Target = 'Monocarboxylate transporter 4'
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610836(MSC-4381)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610833(CHEMBL5276884)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610834(CHEMBL5279064)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610830(CHEMBL5267752)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610837(CHEMBL5281492)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610835(CHEMBL5267349)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610826(CHEMBL5287351)
Affinity DataKi:  29nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610827(CHEMBL5287780)
Affinity DataKi:  32nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610824(CHEMBL5268966)
Affinity DataKi:  37nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610829(CHEMBL5288904)
Affinity DataKi:  51nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610831(CHEMBL5265956)
Affinity DataKi:  56nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610825(CHEMBL5266104)
Affinity DataKi:  99nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610828(CHEMBL5271816)
Affinity DataKi:  222nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Mus musculus)TBA
LigandPNGBDBM50610868(CHEMBL5282978)
Affinity DataKi:  301nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50608641(AF 2838 | AF-2838 | BINDARIT | Bindarit)
Affinity DataKi:  3.02E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356873(US10214492, Example 223 | US11292767, Example 223)
Affinity DataIC50:  0.300nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356873(US10214492, Example 223 | US11292767, Example 223)
Affinity DataIC50:  0.300nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356917(US10214492, Example 268 | US11292767, Example 268)
Affinity DataIC50:  0.300nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356917(US10214492, Example 268 | US11292767, Example 268)
Affinity DataIC50:  0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356917(US10214492, Example 268 | US11292767, Example 268)
Affinity DataIC50:  0.300nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356790(US10214492, Example 155 | US11292767, Example 155)
Affinity DataIC50:  0.320nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356790(US10214492, Example 155 | US11292767, Example 155)
Affinity DataIC50:  0.320nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356906(US10214492, Example 257 | US11292767, Example 257)
Affinity DataIC50:  0.350nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356913(US10214492, Example 264)
Affinity DataIC50:  0.350nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356906(US10214492, Example 257 | US11292767, Example 257)
Affinity DataIC50:  0.350nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM546758((2R)-2-([5-(3,5-Dimethoxyphenyl)-1- [(2-ethoxyphen...)
Affinity DataIC50:  0.350nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356915(US10214492, Example 266 | US11292767, Example 266)
Affinity DataIC50:  0.360nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356915(US10214492, Example 266 | US11292767, Example 266)
Affinity DataIC50:  0.360nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356915(US10214492, Example 266 | US11292767, Example 266)
Affinity DataIC50:  0.360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356870(US10214492, Example 220 | US11292767, Example 220)
Affinity DataIC50:  0.540nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356870(US10214492, Example 220 | US11292767, Example 220)
Affinity DataIC50:  0.540nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356916(US10214492, Example 267 | US11292767, Example 267)
Affinity DataIC50:  0.570nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356916(US10214492, Example 267 | US11292767, Example 267)
Affinity DataIC50:  0.570nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356916(US10214492, Example 267 | US11292767, Example 267)
Affinity DataIC50:  0.570nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356805(US10214492, Example 167 | US11292767, Example 167)
Affinity DataIC50:  0.590nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356805(US10214492, Example 167 | US11292767, Example 167)
Affinity DataIC50:  0.590nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356811(US10214492, Example 172 | US11292767, Example 172)
Affinity DataIC50:  0.590nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356811(US10214492, Example 172 | US11292767, Example 172)
Affinity DataIC50:  0.590nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356909(US10214492, Example 260 | US11292767, Example 260)
Affinity DataIC50:  0.830nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356909(US10214492, Example 260 | US11292767, Example 260)
Affinity DataIC50:  0.830nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356918(US10214492, Example 269 | US11292767, Example 269)
Affinity DataIC50:  1nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM345281(2-[[1-[(2-Chlorophenyl)methyl]-5-(3- isobutoxyphe...)
Affinity DataIC50:  1nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356918(US10214492, Example 269 | US11292767, Example 269)
Affinity DataIC50:  1nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50606665(Isotense | Londomin | NSC-77030 | Neoreserpan | SU...)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50606664(CHEMBL1616099)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM345281(2-[[1-[(2-Chlorophenyl)methyl]-5-(3- isobutoxyphe...)
Affinity DataIC50:  1nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50606665(Isotense | Londomin | NSC-77030 | Neoreserpan | SU...)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human NCI-H358 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM345281(2-[[1-[(2-Chlorophenyl)methyl]-5-(3- isobutoxyphe...)
Affinity DataIC50:  1nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM345281(2-[[1-[(2-Chlorophenyl)methyl]-5-(3- isobutoxyphe...)
Affinity DataIC50:  1nMAssay Description:MDA-MB-231 breast cancer cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50606664(CHEMBL1616099)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human NCI-H358 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
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