Compile Data Set for Download or QSAR
maximum 50k data
Found 187 of kd for UniProtKB: P19793
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKd:  13nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  36nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  7nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  26nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  42nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKd:  40nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKd:  30nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  51nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
TargetDimer of Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  28nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
TargetDimer of Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  18nMpH: 7.4 T: 2°CAssay Description:Binding assay using human retinoid X receptor alpha (RXR).More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKd:  9nMAssay Description:Compound was tested for binding affinity against retinoid X receptor using 5 nM of [3H]-9-cis-RA as a radioligand in baculovirus expressed receptorMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50122352((2E,4E)-3-Methyl-6-[1-(3,5,5,8,8-pentamethyl-5,6,7...)
Affinity DataKd:  16nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50122350((2E,4E)-3-Methyl-6-[1-(5,5,8,8-tetramethyl-5,6,7,8...)
Affinity DataKd:  41nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50122351((2E,4E)-3-Methyl-6-[1-(5,5,8,8-tetramethyl-5,6,7,8...)
Affinity DataKd:  2nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50122348((2E,4E)-6-[1-(3,5-Di-tert-butyl-phenyl)-cyclopropy...)
Affinity DataKd:  3nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKd:  9nMAssay Description:Relative activity against Retinoid X receptor RXR-alpha compared to 9-cis-RAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040023(4-(3-Fluoro-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro...)
Affinity DataKd:  706nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032667(4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd:  195nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040011(4-(3-Bromo-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-...)
Affinity DataKd:  105nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040021(4-[1-(3-Isopropyl-5,5,8,8-tetramethyl-5,6,7,8-tetr...)
Affinity DataKd:  55nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040017(4-[1-(3-Ethyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahyd...)
Affinity DataKd:  31nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040025(4-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040013(4-(3-Chloro-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro...)
Affinity DataKd:  130nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040015(4-[1-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrah...)
Affinity DataKd:  96nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040014(4-[1-(3-Fluoro-5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataKd:  69nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040024(4-[1-(3-Hydroxy-5,5,8,8-tetramethyl-5,6,7,8-tetrah...)
Affinity DataKd:  487nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040016(4-[1-(3-Chloro-5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataKd:  27nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040012(4-[1-(3-Bromo-5,5,8,8-tetramethyl-5,6,7,8-tetrahyd...)
Affinity DataKd:  28nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataKd: >200nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032677(4-[1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-nap...)
Affinity DataKd:  110nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032672(4-[1-(3,8,8-Trimethyl-5,6,7,8-tetrahydro-naphthale...)
Affinity DataKd: >1.00E+3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd:  36nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032674(4-[2-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-nap...)
Affinity DataKd:  670nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032667(4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd:  138nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032664(4-[1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-nap...)
Affinity DataKd:  46nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032665(4-[1-(3,5,5-Trimethyl-5,6,7,8-tetrahydro-naphthale...)
Affinity DataKd:  1.16E+3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032662(4-[1-(1,1,2,3,3,6-Hexamethyl-indan-5-yl)-vinyl]-be...)
Affinity DataKd:  176nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032663(4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd: >1.00E+3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032668(4-[2-Methyl-1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetra...)
Affinity DataKd:  50nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032676(4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd:  520nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032673(2-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd: >1.00E+3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032670(4-[1-Methyl-1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetra...)
Affinity DataKd: >1.00E+3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032669(3-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd: >1.00E+3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032666(6-[1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-nap...)
Affinity DataKd:  22nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50032671(6-[1-(3,5,5,8,8-PENTAMETHYL-5,6,7,8-TETRAHYDRONAPH...)
Affinity DataKd:  3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataKd:  3nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataKd:  16nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataKd: >200nMAssay Description:Binding affinity for human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKd: >200nMAssay Description:Inhibition of binding to human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University of Texas Southwestern Medical Center

LigandPNGBDBM50040020(4-[1-(5,5,8,8-Tetramethyl-3-propyl-5,6,7,8-tetrahy...)
Affinity DataKd:  137nMAssay Description:Inhibition of [3H]-9-cis-RA binding to baculovirus expressed retinoid receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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