Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 2 of ec50 for monomerid = 50106297
TargetNuclear receptor ROR-gamma [262-507](Human)
Genentech

US Patent
LigandPNGBDBM50106297(CHEMBL3596274 | US9550771, Example 88)
Affinity DataEC50:  250nMT: 25°CAssay Description:ssays were carried out in 16-μL reaction volumes in black 384 Plus F Proxiplates (Perkin-Elmer 6008269). All assay components except test ligand...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetNuclear receptor ROR-gamma(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50106297(CHEMBL3596274 | US9550771, Example 88)
Affinity DataEC50:  250nMAssay Description:Inverse agonist activity at N-terminal 6xHis-tagged human RORc ligand binding domain (241 to 486) expressed in bacterial expression system assessed a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed