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Report error Found 4 of ic50 for monomerid = 187104
TargetPlasma kallikrein(Human)
Kalvista Pharmceuticals

US Patent
LigandPNGBDBM187104(US9670157, 118 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-...)
Affinity DataIC50:  1nMAssay Description:Plasma kallikrein inhibitory activity in vitro was determined using standard published methods (see e.g. Johansen et al., Int. J. Tiss. Reac. 1986, 8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetPlasma kallikrein(Human)
Kalvista Pharmceuticals

US Patent
LigandPNGBDBM187104(US9670157, 118 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-...)
Affinity DataIC50:  1nMAssay Description:Plasma kallikrein inhibitory activity in vitro was determined using standard published methods (see e.g. Johansen et al., Int. J. Tiss. Reac. 1986, 8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetKallikrein-1(Human)
Kalvista Pharmceuticals

US Patent
LigandPNGBDBM187104(US9670157, 118 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:KLK1 inhibitory activity in vitro was determined using standard published methods (see e.g. Johansen et al., Int. J. Tiss. Reac. 1986, 8, 185; Shori ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetKallikrein-1(Human)
Kalvista Pharmceuticals

US Patent
LigandPNGBDBM187104(US9670157, 118 1-[4-(4-Methyl-pyrazol-1-ylmethyl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:KLK1 inhibitory activity in vitro was determined using standard published methods (see e.g. Johansen et al., Int. J. Tiss. Reac. 1986, 8, 185; Shori ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent