TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity for 5-HT3 receptor of NG108-15 cells using [3H]-GR-65,630More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity towards Opioid receptor kappa 1 by the displacement of [125I]-(D-Pro10)-Dynorphin AMore data for this Ligand-Target Pair
Affinity DataIC50: 248nMAssay Description:Binding affinity towards Opioid receptor delta 1 by the displacement of [125I]-DeltorphinMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of [125I]-Deltorphin binding to human delta opioid receptor from membranes of HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of [125I]-(D-Pro10)-Dynorphin A binding to human kappa opioid receptor from membranes of HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.84E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [125I]Enkephalin; Not determinedMore data for this Ligand-Target Pair