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Report error Found 6 of ic50 for monomerid = 242743
TargetNeuromedin-K receptor(Human)
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US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataIC50:  30nMAssay Description:Chinese Hamster Ovary recombinant cells expressing the human NK-3 receptor and a construct that encodes the photoprotein apoaequorin were used for th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Euroscreen

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataIC50:  30nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Euroscreen

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataIC50:  30nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataIC50:  4.50E+4nMAssay Description:The human ether-a-go-go related gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataIC50:  4.50E+4nMAssay Description:The human ether-a-go-go related gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (Igr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataIC50:  4.50E+4nMAssay Description:The hERG inhibition study aims at quantifying the in vitro effects of compounds of the invention on the potassium-selective IKr current generated in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent