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Found 1 of ic50 for monomerid = 28400
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM28400((2E)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2...)
Affinity DataIC50:  1.20E+3nMpH: 7.5 T: 2°CAssay Description:The activity of Pim kinase was measured in a homogeneous luciferase assay using GST-Pim, biotinylated peptide substrate and a luciferin-luciferase de...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed