Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 50120516
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50120516((7-{[4-(Pyridin-2-ylamino)-butyrylamino]-methyl}-6...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of fibrinogen from Human integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50120516((7-{[4-(Pyridin-2-ylamino)-butyrylamino]-methyl}-6...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at alphavbeta5 integrin receptor (unknown origin) by cell-free ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50120516((7-{[4-(Pyridin-2-ylamino)-butyrylamino]-methyl}-6...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of fibrinogen from Human integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50120516((7-{[4-(Pyridin-2-ylamino)-butyrylamino]-methyl}-6...)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor (unknown origin) by cell-free ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50120516((7-{[4-(Pyridin-2-ylamino)-butyrylamino]-methyl}-6...)
Affinity DataIC50:  4.36E+3nMAssay Description:Displacement of vitronectin from human integrin alphaV-beta5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed