Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ic50 for monomerid = 50142759
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50142759((R)-N-(4-(1-(3-(4-tert-butylbenzyl)thioureido)ethy...)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50142759((R)-N-(4-(1-(3-(4-tert-butylbenzyl)thioureido)ethy...)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at TRPV1 in Sprague-Dawley rat DRG neuron assessed as reduction of capsaicin-stimulated intracellular 45Ca2+ influx by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed