Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 2 of ic50 for monomerid = 50216402
TargetP2X purinoceptor 7(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50216402(CHEMBL230925 | N-(2-(4-(4-nitrophenyl)piperazin-1-...)
Affinity DataIC50:  19.9nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as inhibition of BzATP-induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50216402(CHEMBL230925 | N-(2-(4-(4-nitrophenyl)piperazin-1-...)
Affinity DataIC50:  21nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as effect on intracellular calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed