Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 2 of ic50 for monomerid = 50310932
TargetAdenosine receptor A2b(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50310932((+/-)-[2-(1-Pyridin-3-yl-ethylamino)-thieno[3,2-d]...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human adeosine A2B receptor expressed in CHOK1 cells assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50310932((+/-)-[2-(1-Pyridin-3-yl-ethylamino)-thieno[3,2-d]...)
Affinity DataIC50:  2.35E+3nMAssay Description:Antagonist activity at human adeosine A2A receptor expressed in CHOK1 cells assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed