Affinity DataIC50: 25nMAssay Description:Inhibition of CDK2 in presence of 60 uM ATPMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK5/p25 assessed as [33P]gamma-ATP incorporation into peptide PKTPKKAKKL substrate after 45 mins by scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of GSK3beta in presence of 60 uM ATPMore data for this Ligand-Target Pair