Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50343660
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50343660(4-((3,5-diamino-1H-pyrazol-4-yl)diazenyl)benzenesu...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of RSK2 after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Egyptian Russian University

Curated by ChEMBL
LigandPNGBDBM50343660(4-((3,5-diamino-1H-pyrazol-4-yl)diazenyl)benzenesu...)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of human full-length N-terminal GST/His6-tagged CDK9 (1 to 372 residues)/His6-tagged Cyclin-T1 (1 to 726 residues) expressed in sf9 cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Egyptian Russian University

Curated by ChEMBL
LigandPNGBDBM50343660(4-((3,5-diamino-1H-pyrazol-4-yl)diazenyl)benzenesu...)
Affinity DataIC50:  4.17E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected Sf21 insect cells using histone H1 as substrate in presence of [gamma3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed