TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Dr. Reddy'S Laboratories, Ameerpet, Hyderabad, India.
Curated by ChEMBL
Dr. Reddy'S Laboratories, Ameerpet, Hyderabad, India.
Curated by ChEMBL
Affinity DataIC50: 327nMAssay Description:Inhibition of CDK5/p25 assessed as [33P]gamma-ATP incorporation into biotinylated PKTPKKAKKL substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair