TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Normandy University
Curated by ChEMBL
Normandy University
Curated by ChEMBL
Affinity DataIC50: 579nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair