Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 50535009
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50535009(CHEMBL4476840)
Affinity DataIC50:  66nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in baculovirus expression system by kinase-glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50535009(CHEMBL4476840)
Affinity DataIC50:  98nMAssay Description:Inhibition of PI3Kalpha (unknown origin) expressed in baculovirus expression system by kinase-glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50535009(CHEMBL4476840)
Affinity DataIC50:  171nMAssay Description:Inhibition of PI3Kdelta N836D mutant (unknown origin) expressed in Sf21 cells co-expressing p85 by kinase-glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50535009(CHEMBL4476840)
Affinity DataIC50:  329nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in baculovirus expression system by kinase-glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50535009(CHEMBL4476840)
Affinity DataIC50:  496nMAssay Description:Inhibition of PI3Kgamma (unknown origin) expressed in baculovirus expression system by kinase-glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed