Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ic50 for monomerid = 572069
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50:  550nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50:  550nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50:  550nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50:  5.50E+3nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent