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Report error Found 16 of ki for monomerid = 242743
TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  24nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist3 H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  24nMAssay Description:Human NK-3: The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  24nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist3 H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  24nMpH: 7.4Assay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  24nMpH: 7.4Assay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  24nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nMAssay Description:Human NK-1: The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nM ΔG°:  -26.6kJ/molepH: 7.4 T: 25°CAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nM ΔG°:  -26.6kJ/molepH: 7.4 T: 25°CAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nMAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nMAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.50E+4nMAssay Description:The affinity of compounds of the invention for the NK-2 receptor was evaluated in CHO recombinant cells which express the human NK-2 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.50E+4nM ΔG°:  -26.3kJ/molepH: 7.4 T: 25°CAssay Description:The affinity of compounds of the invention for the NK-2 receptor was evaluated in CHO recombinant cells which express the human NK-2 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.50E+4nMAssay Description:The affinity of compounds of the invention for the NK-2 receptor was evaluated in CHO recombinant cells which express the human NK-2 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.50E+4nM ΔG°:  -26.3kJ/molepH: 7.4 T: 25°CAssay Description:The affinity of compounds of the invention for the NK-2 receptor was evaluated in CHO recombinant cells which express the human NK-2 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-K receptor(Human)
Ogeda

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.50E+4nMAssay Description:Human NK-2 The affinity of compounds of the invention for the NK-2 receptor was evaluated in CHO recombinant cells which express the human NK-2 recep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent