Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 8 of ki for monomerid = 50312966
TargetAdenosine receptor A2b(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  239nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in human HeLa cells after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  239nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in human HeLa cells after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  931nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  931nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  3.75E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells after 3 hrs by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50312966(CHEMBL1081971 | N-(6-(furan-2-yl)-5-(pyrimidin-4-y...)
Affinity DataKi:  3.75E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells after 3 hrs by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed