Compile Data Set for Download or QSAR
maximum 50k data
Found 15 of ki for monomerid = 85775
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  108nMAssay Description:Inhibition of [125I]- AB-MECA binding to human Adenosine A3 receptors expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  108nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  108nMAssay Description:Displacement of [125]AB-MECA binding to human Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  110nMAssay Description:Displacement of [125 I]AB-MECA from Adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Chick)
University of Illinois At Chicago

Curated by PDSP Ki Database
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  990nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Chick)
University of Illinois At Chicago

Curated by PDSP Ki Database
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  3.43E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  4.16E+3nMAssay Description:Binding affinity against rat Adenosine A3 receptor from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  4.77E+3nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at Adenosine A2A receptor in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  4.77E+3nMAssay Description:Displacement of [3H]-CGS-21,680 from Adenosine A2A receptor of rat striatal membrane at 10e-4 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  4.77E+3nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  4.77E+3nMAssay Description:Displacement of [3H]-CGS- 21680 binding to Adenosine A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  5.93E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat cerebral cortex membrane by radioligand binding assay using [3H](R)-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  5.93E+3nMAssay Description:Displacement of specific [3H]-(R)-PIA binding at adenosine A1 receptor from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  5.93E+3nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM85775(CHEMBL315984 | MRS1097)
Affinity DataKi:  5.93E+3nMAssay Description:Displacement of [3H](R)-PIA binding to Adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed