Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ki for monomerid = 92862
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Pfizer

LigandPNGBDBM92862(US9284315, BEZ-235 | mTOR Inhibitor, BEZ235)
Affinity DataKi:  1.70nM ΔG°:  -50.1kJ/mole IC50:  3.90nMT: 2°CAssay Description:The LanthaScreen TR-FRET mTOR assay was performed using Costar low-binding 284-well plates at room temperature according to the instructions of the m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Pfizer

LigandPNGBDBM92862(US9284315, BEZ-235 | mTOR Inhibitor, BEZ235)
Affinity DataKi:  2.5nM IC50:  9.60nMAssay Description:The mTOR activity was determined by measuring the amount of [gamma-33 P] phosphae from ATP incorporated in the substrate protein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed