Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 10976
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581757(US11512087, Example 1)
Affinity DataIC50:  2.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581831(US11512087, Example 13-1)
Affinity DataIC50:  3.30nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581837(US11512087, Example 25)
Affinity DataIC50:  3.40nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581838(US11512087, Example 26-1)
Affinity DataIC50:  3.70nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581832(US11512087, Example 13-9)
Affinity DataIC50:  4.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581795(US11512087, Example 4-1)
Affinity DataIC50:  5.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581830(US11512087, Example 12)
Affinity DataIC50:  5.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581780(US11512087, Example 2)
Affinity DataIC50:  5.40nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581829(US11512087, Example 10)
Affinity DataIC50:  6.90nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581828(US11512087, Example 8)
Affinity DataIC50:  7.60nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581835(US11512087, Example 18-1)
Affinity DataIC50:  7.70nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581806(US11512087, Example 4-3)
Affinity DataIC50:  8.5nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581805(US11512087, Example 4-2)
Affinity DataIC50:  9.30nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581836(US11512087, Example 23)
Affinity DataIC50:  9.70nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581833(US11512087, Example 14-4)
Affinity DataIC50:  12nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581834(US11512087, Example 14-11)
Affinity DataIC50:  50nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581806(US11512087, Example 4-3)
Affinity DataIC50:  2.50E+3nMAssay Description:Tyrosine phosphorylation of Lck was performed by using Z′-LYTE Kinase Assay Kit-Tyr 2 Peptide (Invitrogen) containing the following reagents (T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581831(US11512087, Example 13-1)
Affinity DataIC50: >1.00E+4nMAssay Description:Tyrosine phosphorylation of Lck was performed by using Z′-LYTE Kinase Assay Kit-Tyr 2 Peptide (Invitrogen) containing the following reagents (T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM581757(US11512087, Example 1)
Affinity DataIC50: >1.00E+4nMAssay Description:Tyrosine phosphorylation of Lck was performed by using Z′-LYTE Kinase Assay Kit-Tyr 2 Peptide (Invitrogen) containing the following reagents (T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent