Compile Data Set for Download or QSAR
maximum 50k data
Found 114 Enz. Inhib. hit(s) with all data for entry = 11281
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604879(N-(5-Cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-...)
Affinity DataIC50:  0.400nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604880(N-(5-Cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-...)
Affinity DataIC50:  0.600nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604845(N-(5-Cyano-4-(((trans)-2-methoxycyclopentyl)amino)...)
Affinity DataIC50:  0.800nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509949(CHEMBL4475216 | US11667631, Example 29)
Affinity DataIC50:  0.960nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604926(N-(5-Cyano-4-(((trans)-4-methoxytetrahydrofuran-3-...)
Affinity DataIC50:  0.970nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509963(CHEMBL4439119 | US11667631, Example 60)
Affinity DataIC50:  0.990nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604921(N-(5-Cyano-4-trans-((1,2)-2-methoxycyclobutoxy)pyr...)
Affinity DataIC50:  1.02nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604897(N-(5-Cyano-4-(((trans)-4-methoxytetrahydrofuran-3-...)
Affinity DataIC50:  1.12nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509969(CHEMBL4562284 | US11667631, Example 34)
Affinity DataIC50:  1.27nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604909((R)-N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin...)
Affinity DataIC50:  1.28nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604912((R)-N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin...)
Affinity DataIC50:  1.33nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604930(N-(5-Cyano-4-(((3,4)-trans-4-methoxytetrahydro-2H-...)
Affinity DataIC50:  1.34nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509962(CHEMBL4532389 | US11667631, Example 33)
Affinity DataIC50:  1.44nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604924((R)-N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin...)
Affinity DataIC50:  1.62nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604925(N-(5-Cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-...)
Affinity DataIC50:  1.62nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604887(N-(5-Cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-...)
Affinity DataIC50:  1.71nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604883(N-(5-Cyano-4-((1-(methoxymethyl))cyclopropyl)amino...)
Affinity DataIC50:  1.77nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604888(N-(5-Cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-...)
Affinity DataIC50:  2.06nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509951(CHEMBL4446464 | US11667631, Example 35)
Affinity DataIC50:  2.06nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604922(N-(5-Cyano-4-cis-((1,2)-2-methoxycyclobutoxy)pyrid...)
Affinity DataIC50:  2.10nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604902((R)-N-(5-Cyano-4-((1-methoxypropan-2-yl)oxy)pyridi...)
Affinity DataIC50:  2.30nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604927(N-(5-Cyano-4-(((3,4)-trans-4-methoxytetrahydrofura...)
Affinity DataIC50:  2.31nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604923((S)-N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin...)
Affinity DataIC50:  2.49nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604890((S)-N-(5-Cyano-4-((1-methoxypropan-2-yl)amino)pyri...)
Affinity DataIC50:  2.5nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604928(N-(5-Cyano-4-(((3,4)-trans-4-methoxytetrahydro-2H-...)
Affinity DataIC50:  2.73nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604914(N-(5-Cyano-4-(methoxyamino)pyridin-2-yl)-7-formyl-...)
Affinity DataIC50:  2.77nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604891((R)-N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin...)
Affinity DataIC50:  2.89nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604846(N-(5-Cyano-4-((2-(pyrrolidin-1-yl)ethyl)amino)pyri...)
Affinity DataIC50:  2.90nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604906(N-(5-Cyano-4-trans-(((3,4)-4-methoxytetrahydrofura...)
Affinity DataIC50:  2.93nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604892((S)-N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin...)
Affinity DataIC50:  3.15nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509961(CHEMBL4469046 | US11667631, Example 39)
Affinity DataIC50:  3.27nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604928(N-(5-Cyano-4-(((3,4)-trans-4-methoxytetrahydro-2H-...)
Affinity DataIC50:  3.30nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604881(N-(5-Cyano-4-((2-methoxyphenyl)amino)pyridin-2-yl)...)
Affinity DataIC50:  3.40nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509958(CHEMBL4571626 | US11667631, Example 51)
Affinity DataIC50:  3.46nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604885(N-(5-Cyano-4-(((cis)-2-methoxycyclopentyl)amino)py...)
Affinity DataIC50:  3.69nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509968(CHEMBL4533002 | US11667631, Example 58)
Affinity DataIC50:  3.78nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604910((S)-N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin...)
Affinity DataIC50:  3.86nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604896((S)-N-(5-Cyano-4-((tetrahydrofuran-2-yl)thio)pyrid...)
Affinity DataIC50:  4.25nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604903(N-(5-Cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-...)
Affinity DataIC50:  4.41nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604886(N-(5-Cyano-4-(((trans)-2-methoxycyclopentyl)oxy)py...)
Affinity DataIC50:  4.57nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509966(CHEMBL4587476 | US11667631, Example 13)
Affinity DataIC50:  4.61nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509960(CHEMBL4564505 | US11667631, Example 38)
Affinity DataIC50:  4.65nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604905(N-(5-Cyano-4-(((S)-tetrahydrofuran-3-yl)thio)pyrid...)
Affinity DataIC50:  4.66nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604919(N-(5-Cyano-4-(((1S,2S)-2-methoxycyclopentyl)amino)...)
Affinity DataIC50:  4.67nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509972(CHEMBL4470137 | US11667631, Example 41)
Affinity DataIC50:  4.69nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604882(N-(5-Cyano-4-(((1-methoxycyclopropyl)methyl)amino)...)
Affinity DataIC50:  4.70nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604907(N-(5-Cyano-4-(((3,4)-trans-4-methoxytetrahydrofura...)
Affinity DataIC50:  4.95nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604848(N-(5-Cyano-4-(3-methoxypyrrolidin-1-yl)pyridin-2-y...)
Affinity DataIC50:  5.10nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM50509964(CHEMBL4472588 | US11667631, Example 55)
Affinity DataIC50:  5.29nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jiangsu Hansoh Pharmaceutical Group

US Patent
LigandPNGBDBM604847(N-(5-Cyano-4-((2-methyltetrahydrofuran-3-yl)thio)p...)
Affinity DataIC50:  5.40nMAssay Description:In this experiment, the inhibitory effect of the compounds on FGFR4 kinase activity was tested by a fluorescence resonance energy transfer (TR-FRET) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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